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产品信息
Peptide Sequence Z-Gly-Pro-Phe-Leu-CHO
Form White lyophilized solid
Primary Target branched chain amino acid preferring,small neutral amino acid preferring, chymotrypsin-like activities
Primary Target Ki 1.5 , 2.3 , and 40.5 µM
Secondary target IC50 = 3.1 µM for peptidyl-glutamyl peptide hydrolyzing activity
Protect from Light 是的
Packaged under inert gas 是的
Purity ≥90% by HPLC
Chemical formula C30H38N4O6
Storage -20°C
A tetrapeptide aldehyde that acts as a highly selective and potent proteasomal inhibitor (Ki = 1.5 µM for branched chain amino acid preferring, 2.3 µM for small neutral amino acid preferring, and 40.5 µM for chymotrypsin-like activities; IC50 = 3.1 µM for peptidyl-glutamyl peptide hydrolyzing activity). Shown to be a weak inhibitor of trypsin-like proteasomal activity. |