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Zaprinast
A PDE V inhibitor
Product Overview
Product Name: Zaprinast
Alternate Name/Synonyms: 1,4-Dihydro-5-(2-propoxyphenyl)-7H-1,2,3-triazolo(4,5-d)pyrimidin-7-one; M&B 22948
Description: Cell-permeable. A selective inhibitor of cGMP-specific phosphodiesterase (PDE V) (IC₅₀ = 0.45 µM). Inhibits PDE IX only at higher concentrations (IC₅₀ = 35 µM).
Peptide Sequence: N/A
Appearance: White solid
Formulation: N/A
CAS Number: 37762-06-4
Molecular Formula: C₁₃H₁₃N₅O₂
Molecular Weight: 271.27
Purity: ≥98% by HPLC
Solubility:DMSO (100 mM)
Storage Temp.: RT
Shipping Conditions: RT
Handling: Protect from air and light
SMILES: CCCOC1=CC=CC=C1C2=NC(=O)C3=NNNC3=N2
InChi: InChI=1S/C13H13N5O2/c1-2-7-20-9-6-4-3-5-8(9)11-14-12-10(13(19)15-11)16-18-17-12/h3-6H,2,7H2,1H3,(H2,14,15,16,17,18,19)
InChi Key: REZGGXNDEMKIQB-UHFFFAOYSA-N
PubChem CID: 5722
MDL Number: MFCD00214073
USAGE: For Research Use Only! Not For Use in Humans. |