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P-GLYCOPROTEIN INHIBITOR, C-4

产品编号: 517301-10MG     查看说明书
产品名称: P-GLYCOPROTEIN INHIBITOR, C-4  .0   订购此产品 
供应商: Merck
规格: ***
目录价: 2141
库存状态: 3周到货
CAS编号:
应用范围: 生化实验
种属来源:
相关信息:

P-Glycoprotein Inhibitor, C-4
(E)-4-Chloro-N-(3-(3-(4-hydroxy-3-methoxyphenyl)acryloyl)phenyl)benzamide, C-4
A cell-permeable cinnamoyl compound that reversibly inhibits P-gp (P-glycoprotein) efflux function and reverses the MDR (multidrug resistance) phenotype with no noticeable effect on P-gp expression. Shown to significantly enhance Paclitaxel- (Cat. No. 580555) and Vincristine- (Cat. No. 677181) induced cytotoxicity as well as apoptosis in P-gp expressing KBV20C cells.
产品信息
Form  Yellow solid
Molar mass  407.9
Protect from Light  是的
Packaged under inert gas  是的
Purity  ≥95% by HPLC
Solubility  DMSO
Chemical formula  C23H18ClNO4
商店和运输信息
Storage  +2°C to +8°C
Ship  Ambient Temperature Only
Standard Handling

保存条件: 2°C - 8°C
说明书地址: 点击查看详细
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