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PD 145065
A highly potent but non-selective endothelin receptor antagonist [IC50 = 4 nM for the ETA receptor (rabbit renal artery vascular smooth muscle cells); IC50 = 15 nM for the ETB receptor (rat cerebellum)].
产品信息
Peptide Sequence Ac-D-Bhg-Leu-Asp-Ile-Ile-Trp-OH (Bhg = 5H-dibenzo[a,d]cycloheptene-5-glycine)
Form White solid
Molar mass 992.1
Purity ≥98% by HPLC
Solubility Phosphate Buffer, pH 7.5
Chemical formula C52H63N7O10 · 2Na
CAS number 153049-49-1
商店和运输信息
Storage +2°C to +8°C
Ship Ambient Temperature Only
Standard Handling |