BQ-610 A highly selective ETA receptor antagonist (IC50 = 20 nM) that attenuates ET-induced reduction in cardiac output. Also inhibits ET-1- and ET-3-induced activation of adenylate cyclase (IC50 = 28.2 nM). BQ-610 is 30-fold more potent than BQ-123 (Cat. No. 05-23-3831) in porcine aortic smooth muscle membrane assay. 产品信息 Peptide Sequence Homopiperidinyl-CO-Leu-D-Trp(CHO)-D-Trp-ONH4 Form White lyophilized powder Formulation Supplied as an ammonium salt. Molar mass 673.8 Hygrocopic 是的 Purity ≥90% by HPLC Solubility H2O Chemical formula C36H47N7O6 商店和运输信息 Storage -20°C Ship Ambient Temperature Only Standard Handling